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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 28-abr-2016 | Genomic and Molecular Characterization of Miltefosine Resistance in Leishmania infantum Strains with Either Natural or Acquired Resistance through Experimental Selection of Intracellular Amastigotes | Mondelaers, Annelies; Sánchez-Cañete, María P.; Hendrickx, Sarah; Eberhardt, Eline; García-Hernández, Raquel CSIC ORCID; Lachaud, Laurence; Cotton, James; Sanders, Mandy; Cuypers, Bart; Imamura, Hideo; Dujardin, J. C.; Delputte, Peter; Cos, Paul; Caljon, Guy; Gamarro, Francisco; Castanys, Santiago; Maes, Louis | artículo |
closedAccess | | 2001 | High-affinity binding of silybin derivatives to the nucleotide-binding domain of a Leishmania tropica P-glycoprotein-like transporter and chemosensitization of a multidrug-resistant parasite to daunomycin | Pérez-Victoria, J. M. ; Pérez-Victoria, F. J.; Conseil, G.; Maitrejean, M.; Barron, D.; Castanys, Santiago; Gamarro, Francisco; Di Pietro, A.; Comte, Gilles | artículo |
closedAccess | | 2007 | Inactivation of the miltefosine transporter, LdMT, causes miltefosine resistance that is conferred to the amastigote stage of Leishmania donovani and persists in vivo | Seifert, K.; Pérez-Victoria, F. J.; Stettler, M.; Sánchez-Cañete, María P.; Castanys, Santiago; Gamarro, Francisco; Croft, S.L. | artículo |
closedAccess | | 2011 | Increased glycolytic ATP synthesis is associated with tafenoquine resistance in Leishmania major | Manzano, José Ignacio CSIC ORCID; Carvalho, L.; Pérez-Victoria, J. M. ; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2006 | Insights into the molecular mechanism of action of Celastraceae sesquiterpenes as specific, non-transported inhibitors of human P-glycoprotein | Muñoz-Martínez, F.; Reyes, C. P.; Pérez-Lomas, Antonio L.; Jiménez, I. A.; Gamarro, Francisco; Castanys, Santiago | artículo |
closedAccess | | 1998 | Involvement of thiol metabolism in resistance to glucantime in Leishmania tropica | Arana, F. E.; Pérez-Victoria, J. M. ; Repetto, Y.; Morello, A.; Castanys, Santiago; Gamarro, Francisco | artículo |
openAccess | | 2013 | LABCG2, a New ABC Transporter Implicated in Phosphatidylserine Exposure, Is Involved in the Infectivity and Pathogenicity of Leishmania | Campos-Salinas, Jenny; León-Guerrero, D.; González-Rey, Elena CSIC ORCID; Delgado, M.; Castanys, Santiago; Pérez-Victoria, J. M. ; Gamarro, Francisco | artículo |
openAccess | | 2012 | Leishmania donovani Develops Resistance to Drug Combinations | García-Hernández, Raquel CSIC ORCID; Manzano, José Ignacio CSIC ORCID; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2003 | Leishmania donovani resistance to miltefosine involves a defective inward translocation of the drug | Pérez-Victoria, F. J.; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2011 | Leishmanicidal and reversal multidrug resistance constituents from Aeonium lindleyi | Kennedy, M. L.; Cortés, Fernando; Piñero, J. E.; Castanys, Santiago; López-Arencibia, A.; Gamarro, Francisco; Bazzocchi, I. L.; Jiménez, I. A. | artículo |
closedAccess | | 2009 | Low plasma membrane expression of the miltefosine transport complex renders leishmania braziliensis refractory to the drug | Sánchez-Cañete, María P.; Carvalho, L.; Pérez-Victoria, F. J.; Gamarro, Francisco; Castanys, Santiago | artículo |
closedAccess | | 2006 | Mechanisms of experimental resistance of Leishmania to miltefosine: Implications for clinical use | Pérez-Victoria, F. J.; Sánchez-Cañete, María P.; Seifert, K.; Croft, S.L.; Sundar, S.; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 1999 | New natural sesquiterpenes as modulators of daunomycin resistance in a multidrug-resistant Leishmania tropica line | Pérez-Victoria, J. M. ; Tincusi, B. M.; Jiménez, I. A.; Bazzocchi, I. L.; Gupta, M. P.; Castanys, Santiago; Gamarro, Francisco; Ravelo, Ángel G. | artículo |
closedAccess | | 2008 | New terpenoids from Maytenus apurimacensis as MDR reversal agents in the parasite Leishmania | Delgado-Méndez, P.; Herrera, N.; Herrera, N.; Chávez, H.; Estévez-Braun, Ana; Ravelo, Ángel G.; Cortés, Fernando; Castanys, Santiago; Gamarro, Francisco | artículo |
openAccess | | 2011 | Non-reducing trisaccharide fatty acid monoesters: Novel detergents in membrane biochemistry | Pérez-Victoria, Ignacio; Pérez-Victoria, F. J.; Roldán-Vargas; García-Hernández, Raquel CSIC ORCID; Carvalho, Luis; Castanys, Santiago; Gamarro, Francisco; Morales, Juan C.; Pérez-Victoria, J. M. | artículo |
closedAccess | | 2009 | Novel dihydro-β-agarofuran sesquiterpenes as potent modulators of human P-glycoprotein dependent multidrug resistance | Torres-Romero, D.; Muñoz-Martínez, F.; Jiménez, I. A.; Castanys, Santiago; Gamarro, Francisco; Bazzocchi, I. L. | artículo |
closedAccess | | 2012 | Oxazolo[3,2-a]pyridine. A new structural scaffold for the reversal of multi-drug resistance in Leishmania | Caballero, E.; Manzano, José Ignacio CSIC ORCID; Puebla, P.; Castanys, Santiago; Gamarro, Francisco; San Feliciano, A. | artículo |
closedAccess | | 2006 | Phospholipid translocation and miltefosine potency require both L. donovani miltefosine transporter and the new protein LdRos3 in Leishmania parasites | Pérez-Victoria, F. J.; Sánchez-Cañete, María P.; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2003 | Rapid transport of phospholipids across the plasma membrane of Leishmania infantum | Araújo-Santos, J. M.; Gamarro, Francisco; Castanys, Santiago; Herrmann, A.; Pomorski, T. G. | artículo |
openAccess | | 2011 | Reversal of P-Glycoprotein-Mediated Multidrug Resistance by Terpenoids from Maytenus Species | Kennedy, M. L.; Llanos, G. G.; Castanys, Santiago; Gamarro, Francisco; Bazzocchi, I. L.; Jiménez, I. A. | preprint |