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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccessPost-Print-2009-JOC-9071.pdf.jpg2009One-Pot Synthesis of Polycyclic Nucleosides with Unusual Molecular SkeletonsBonache, María-Cruz CSIC; Cordeiro, Alessandra CSIC; Carrero, Paula CSIC; Quesada, Ernesto CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
openAccessAntimicrob. Agents Chemother.-2016-Rivero-Buceta-5064-7.pdf.jpg2016Optimization of a class of tryptophan dendrimers that inhibit HIV replication leads to a selective, specific, and low-nanomolar inhibitor of clinical isolates of enterovirus A71Rivero-Buceta, Eva CSIC ORCID; Sun, L.; Martínez-Gualda, Belén CSIC; Doyagüez, Elisa G. CSIC; Donckers, K.; Quesada, Ernesto CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Delang, Leen; San-Félix, Ana CSIC ORCID ; Neyts, Johan; Leyssen, Pieterartículo
openAccessEuropean Journal of Medicinal Chemistry 237.pdf.jpgabr-2022Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitorsMartí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Fernández-Barahona, Irene; Mills, Alberto; Abdelnabi, Rana; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Herranz, Fernando CSIC ORCID CVN; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
openAccessPeptides Linked to Vpg1.pdf.jpg13-jun-2019Peptides Linked to Vpg1 of Foot-and-Mouth Disease Virus (FMDV): Design, Synthesis and X-Ray Crystallography of the Complexes with FMDV RNA-dependent RNA polymeraseCastro, Sonia de CSIC ORCID; Ferrer-Ortra, C.; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Camarasa Rius, María José CSIC ORCIDcomunicación de congreso
openAccessACSMCL2020_RT-dimeriz-inhibs-3(revised-for publication).pdf.jpg2020Peptides mimicking the β7/β8 loop of HIV'1 reverse transcriptase p51 as “hotspot-targeted” dimerization inhibitorsSánchez-Murcia, Pedro A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-Aparicio, Carlos CSIC; Jiménez, M. Angeles CSIC ORCID ; Corona, A.; Tramontano, Enzo; Sluis-Cremer, N.; Menéndez-Arias, Luis CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCIDartículo
openAccessaccesoRestringido.pdf.jpg2018Polypharmacology in HIV inhibition: can a drug with simultaneous action against two relevant targets be an alternative to combination therapy?Castro, Sonia de CSIC ORCID; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess6-jun-2013Probing the Dimerization Interface of Leishmania infantum Trypanothione Reductase with Site-Directed Mutagenesis and Short PeptidesToro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Moreno, David; Ruiz-Santaquiteria, Marta CSIC ORCID; Alzate, Juan Fernando; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Jiménez-Ruiz, Antonioartículo
openAccessaccesoRestringido.pdf.jpg2018Prodrugs of Nucleoside Triphosphates as a Sound and Challenging Approach: A Pioneering Work That Opens a New Era in the Direct Intracellular Delivery of Nucleoside TriphosphatesCamarasa Rius, María José CSIC ORCIDartículo; preprint
openAccessCA2525191A1.pdf.jpg18-nov-2004Produgs cleavable by CD26.Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNpatente
openAccessProtein ligand complex.pdf.jpg23-ene-2018Protein-ligand complex for structure-based design: impact on the affinity and antitumor activity of new tubulin ligandsBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDcomunicación de congreso
openAccessBrit. J. Pharmacol..pdf.jpg2020Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein–protein interaction disruptorLucio, Héctor de; Toro, Miguel Ángel; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Jimenez-Ruiz, Antonioartículo
openAccessaccesoRestringido.pdf.jpg2019Pyrrolopyrimidine vs imidazole-phenyl-thiazole scaffolds in nonpeptidic dimerization inhibitors of leishmania infantum trypanothione reductaseRevuelto, Alejandro CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Lucio, Héctor de; Gamo, Ana; Carriles, Alejandra A. CSIC ORCID; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccessaccesoRestringido.pdf.jpg2008Reactivity of the 4-amino-5H-1,2-oxathiole-2,2-dioxide heterocyclic system: A combined experimental and theoretical studyCastro, Sonia de CSIC ORCID ; Peromingo, M. T.; Lozano, Ángel E. ; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccess2012Recent Advances in Thymidine Kinase 2 (TK2) Inhibitors and New Perspectives for Potential ApplicationsPriego, Eva María CSIC ORCID; Karlsson, Anna; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessASF9 REVISED jm-2019-01737d.pdf.jpgene-2020Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry InhibitorsMartínez-Gualda, Belén CSIC; Sun, Liang; Martí-Marí, Olaia CSIC ORCID; Abdelnabi, Rana; Noppen, Sam; Bator, Carol M.; Quesada, Ernesto CSIC ORCID ; Delang, Leen; Mirabelli, Carmen; Lee, Hyunwook; Schols, Dominique; Neyts, Johan; Hafenstein, Susan; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2001Second generation of TSAO compounds directed against HIV-1 TSAO-resistant strainsLobaton, E.; Velázquez, Sonsoles CSIC ORCID CVN; Peréz-Pérez, María-Jesús CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; San-Felix, S.; De Clercq, Erik; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2008Selective human adenosine A3 antagonists based on pyrido[2,1-f]purine-2,4-diones: Novel features of hA3 antagonist bindingPriego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Von Frijtag Drabbe Kuenzel, J. K.; de Vries, H.; Ijzerman, A. P.; Camarasa Rius, María José CSIC ORCID; Martín-Santamaría, Sonsoles CSIC ORCID artículo
openAccesspost-Print-2011-AntiviralResearch-37.pdf.jpg2011Selective inhibition of Human Immunodeficiency Virus type 1 (HIV-1) by a novel family of tricyclic nucleosidesBonache, María-Cruz CSIC; Cordeiro, Alessandra CSIC; Quesada, Ernesto CSIC ORCID ; Vanstreels, Els; Daelemans, Dirk; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; San-Félix, Ana CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg1982Síntesis, actividad citostática y mecanismo de acción de N-glicosil-halometilazoles. Un nuevo tipo de agentes alquilantesAlonso, Gregorio; Alonso, R.; Camarasa Rius, María José CSIC ORCID; Contreras, Antonio; García-López, M. Teresa CSIC ; Heras, F. G. de las; Herranz, Rosario CSIC ORCID; Sanchez-Perez, Rosa M.artículo
openAccesspharmaceuticals-14-00689-v2-1.pdf.jpg17-jul-2021Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide ReductaseRevuelto, Alejandro CSIC ORCID; López-Martín, Isabel; Lucio, Héctor de; García-Soriano, Juan Carlos; Zanda, Nicola; Castro, Sonia de CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCIDartículo