Mostrando resultados 25 a 44 de 131
< Anterior
Siguiente >
Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 28-abr-2011 | Derivados de nucleósidos para el tratamiento de infecciones por Leishmania | Gago, Federico CSIC ORCID; Rico Galán, Eva; Camarasa Rius, María José CSIC ORCID; Jiménez, A. R.; Casanova Malpica, Elena; Moreno Mateos, David; Peréz-Pérez, María-Jesús CSIC ORCID | patente |
openAccess | | 2019 | Design and Synthesis of New 6-Nitro and 6-Amino- 3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole Derivatives: Antiproliferative and Antibacterial Activity | Cuartas, Viviana; Crespo, María del Pilar; Priego, Eva María CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 2019 | Design and synthesis of new 6-nitro and 6-Amino-3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole derivatives: Antiproliferative and antibacterial activity | Cuartas, V.; Crespo, M. D. P.; Priego, Eva María CSIC ORCID; Persoons, L.; Daelemans, D.; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 2010 | Design, synthesis and inhibitory activity against Mycobacterium tuberculosis thymidine monophosphate kinase of acyclic nucleoside analogues with a distal imidazoquinolinone | Familiar, Olga CSIC; Munier-Lehmann, Hélène; Aínsa, José A.; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 14-oct-2014 | Design, synthesis and X-Ray of Foot-and-mouth disease virus (Fluoro)uridylylated peptides linked to the genome (VPgpU and VPgpFU) | Castro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Domingo, Esteban CSIC ORCID; Camarasa Rius, María José CSIC ORCID | póster de congreso |
openAccess | | 2015 | Design, synthesis, and biological evaluation of unconventional aminopyrimidine, aminopurine, and amino-1,3,5-triazine methyloxynucleosides | Fernández-Cureses, Gloria CSIC; Castro, Sonia de CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2013 | Differential Recognition of Mannose-Based Polysaccharides by Tripodal Receptors Based on a Triethylbenzene Scaffold Substituted with Trihydroxybenzoyl Moieties | Carrero, Paula CSIC; Ardá, Ana CSIC ORCID CVN; Álvarez-Pérez, Mónica CSIC ORCID; Doyagüez, Elisa G. CSIC; Rivero-Buceta, Eva CSIC ORCID; Quesada, Ernesto CSIC ORCID ; Prieto Orzanco, Alicia CSIC ORCID ; Solís, Dolores; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Jiménez-Barbero, Jesús CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
closedAccess | | 2011 | Dipeptidyl peptidase IV dependent water-soluble prodrugs of highly lipophilic bicyclic nucleoside analogues | Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Andrei, G; Snoeck, R.; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2012 | Dipeptidyl Peptidase IV-Activated Prodrugs of Anti- Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer Systems | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2015 | Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: A successful strategy for improving water solubility and oral bioavailability | Velázquez, Sonsoles CSIC ORCID CVN; Castro, Sonia de CSIC ORCID; Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 3-feb-2012 | Dipeptidyl-peptidase IV (DPPIV/CD26)-based prodrugs of hydroxy-containing drugs | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; Lambeir, Anne-Marie; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | jun-2019 | Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the aT5 loop | Bueno, Oskia CSIC; Gargantilla, Marta CSIC ORCID; Estévez-Gallego, Juan CSIC ORCID ; Martins, Solange; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | artículo |
closedAccess | | 2014 | Discovery and SAR studies of a novel class of cytotoxic 1,4-disubstituted piperidines via Ugi reaction | Castro, Sonia de CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2006 | Discovery of TSAO derivatives with an unusual HIV-1 activity/resistance profile | Castro, Sonia de CSIC ORCID ; García-Aparicio, Carlos CSIC; Van Laethem, K.; Gago, Federico CSIC ORCID; Lobatón, E.; De Clercq, E.; Balzarini, J.; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2014 | Diseño y desarrollo de una novedosa estrategia profármaco basada en la enzima DPPIV/CD26 | Camarasa Rius, María José CSIC ORCID; Castro, Sonia de CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 7-jul-2021 | Double Arylation of the Indole Side Chain of Tri- and Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV‑1 and EV-A71 Entry Inhibitors | Martí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Puente-Secades, Sofía de la CSIC; Mills, Alberto; Quesada, Ernesto CSIC ORCID ; Abdelnabi, Rana; Sun, Liang; Boonen, Arnaud; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | 2021 | Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazoles | Revuelto, Alejandro CSIC ORCID; Lucio, Héctor de; García-Soriano, Juan Carlos; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2012 | Efficient synthesis and anti-enteroviral activity of 9-arylpurines | Aguado, Leire CSIC; Canela, María-Dolores CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Leyssen, Pieter; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 2019 | Enzymatic and Chemical Synthesis of Nucleic Acid Derivatives | Camarasa Rius, María José CSIC ORCID; Fernandez Lucas, Jesús | libro |
closedAccess | | 2008 | Exploring acyclic nucleoside analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase | Familiar, Olga CSIC; Munier-Lehmann, Hélène; Negri, Ana; Gago, Federico CSIC ORCID; Douguet, D.; Rigouts, L.; Hernández, A. -I.; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |