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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
closedAccessaccesoRestringido.pdf.jpg2013A fluorescent styrylquinoline with combined therapeutic and diagnostic activities against Alzheimer's and prion diseasesStaderini, Matteo; Aulic, Suzana; Bartolini, Manuela; Tran, H. N. A.; González-Ruiz, Victor; Pérez, Daniel I. CSIC ORCID; Cabezas, Nieves; Martínez Gil, Ana CSIC ORCID ; Martín, M. Antonia; Andrisano, Vincenza; Legname, Giuseppe; Menéndez, José Carlos; Bolognesi, Maria Lauraartículo
openAccessACSChemNeurosci 2018.pdf.jpg9-oct-2018A focused library of psychotropic analogs with neuroprotective and neuroregenerative potentialUliassi, Elisa; Peña-Altamira, Luis Emiliano; Morales, Aixa V. CSIC ORCID; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martínez-González, Loreto CSIC ORCID ; Martínez Gil, Ana CSIC ORCID ; Monti, B.; Bolognesi, Maria Lauraartículo
closedAccessaccesoRestringido.pdf.jpg2012A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: Structure-based design, synthesis, and biological evaluationChiriano, G.; De Simone, A.; Mancini, Francesca; Pérez, Daniel I. CSIC ORCID; Cavalli, A.; Bolognesi, Maria Laura; Legname, G.; Martínez, A.; Andrisano, Vincenza; Carloni, Paolo; Roberti, M.artículo
openAccessEuropean Journal of Medicinal Chemistry_Staderini_2022.pdf.jpg15-nov-2022Bifunctional carbazole derivatives for simultaneous therapy and fluorescence imaging in prion disease murine cell modelsStaderini, Matteo; Vanni, Silvia; Colini Baldeschi, Arianna; Giachin, Gabriele; Zattoni, Marco; Celauro, Luigi; Ferracin, Chiara; Bistaffa, Edoardo; Moda, F.; Pérez, Daniel I. CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Martín, M. Antonia; Martín-Cámara, Olmo; Cores, Ángel; Bianchini, Giulia; Kammerer, Robert; Menéndez, J. Carlos; Legname, G.; Bolognesi, Maria Lauraartículo
openAccessRosini_et_al_2006_postprint.pdf.jpgdic-2006Design, synthesis, and biological evaluation of substituted 2,3-dihydro-1H-cyclopenta[b]quinolin-9-ylamine related compounds as fructose-1,6-bisphosphatase inhibitorsRosini, Michela; Mancini, Francesca; Tarozzi, Andrea; Colizzi, Francesco CSIC ORCID; Andrisano, Vincenza; Bolognesi, Maria Laura; Hrelia, Patrizia; Melchiorre, Carloartículo
openAccessacschemneuro.2c00357.pdf.jpg2022Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's DiseaseGandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janockova, Jana; Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero, Diego; Monti, Barbara; Sabate, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Lauraartículo
closedAccessaccesoRestringido.pdf.jpg2015Multitarget drug discovery for Alzheimer's disease: Triazinones as BACE-1 and GSK-3ß inhibitorsPérez, Daniel I. CSIC ORCID; Pérez Castillo, Ana CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Bolognesi, Maria Laura; Cavalli, Andreaartículo
closedAccessaccesoRestringido.pdf.jpgjun-2014Multitarget ligands and theranostics: Sharpening the medicinal chemistry sword against prion diseasesBongarzone, Salvatore CSIC ORCID; Staderini, Matteo; Bolognesi, Maria Lauraartículo
openAccessaccesoRestringido.pdf.jpg2015Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybridsBenchekroun, Mohamed; Bartolini, Manuela; Egea, Javier; Romero Jódar, Alejandro CSIC ORCID; Soriano, Elena CSIC; Pudlo, M.; Luzet, Vincenza; Andrisano, V.; Jimeno, M. Luisa CSIC ORCID; López, M. G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; Andrés, Lucía de CSIC; Herrera-Arozamena, Clara CSIC ORCID CVN; Monti, B.; Bolognesi, Maria Laura; Rodríguez-Franco, María Isabel CSIC ORCID ; Decker, Michael; Marco-Contelles, José CSIC ORCID; Ismaili, L.artículo
openAccessJ. Med. Chem._Staderini_2019.pdf.jpg14-mar-2019Structure-activity relationships and mechanistic studies of novel mitochondria-targeted, leishmanicidal derivatives of the 4-aminostyrylquinoline scaffoldStaderini, Matteo; Piquero, Marta; Abengozar, M. A. CSIC; Nácher-Vázquez, Montserrat CSIC ORCID; Romanelli, Giulia; López-Alvarado, Pilar; Rivas, Luis CSIC ORCID ; Bolognesi, Maria Laura; Menéndez, J. Carlosartículo
closedAccessaccesoRestringido.pdf.jpg2018Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, asmulti-target-directed ligands for Alzheimer's diseaseChioua, Mourad CSIC ORCID ; Buzzi, Eleonora; Moraleda, Ignacio; Iriepa, Isabel; Maj, Maciej; Wnorowski, Artur; Giovannini, Catia; Tamarin, Anna; Portali, Federica; Ismaili, Lhassane; López-Alvarado, Pilar; Bolognesi, Maria Laura; Jóźwiak, Krzysztof; Menéndez, J. Carlos; Marco-Contelles, José CSIC ORCID; Bartolini, Manuelaartículo
closedAccessaccesoRestringido.pdf.jpg2018Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation InhibitorsGandini, A.; Bartolini, M.; Tedesco, D.; Martínez-González, Loreto CSIC ORCID ; Roca, Carlos CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Zaldívar-Díez, Josefa CSIC ORCID; Pérez, Concepción CSIC ORCID; Zuccheri, G.; Miti, Andrea; Feoli, A.; Castellano, S.; Petralla, Sabrina; Monti, B.; Rossi, M.; Moda, F.; Legname, G.; Martínez Gil, Ana CSIC ORCID ; Bolognesi, Maria Lauraartículo
closedAccessaccesoRestringido.pdf.jpg2013The bivalent ligand approach as a tool for improving the in vitro anti-alzheimer multitarget profile of dimebonRosini, M.; Simoni, E.; Bartolini, Manuela; Soriano, Elena CSIC; Marco-Contelles, José CSIC ORCID; Andrisano, V.; Monti, B.; Windisch, M.; Hutter-Paier, B.; McClymont, D. W.; Mellor, I. R.; Bolognesi, Maria Lauraartículo