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| Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
| closedAccess | | 1998 | Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptase | Velázquez, Sonsoles CSIC ORCID CVN; Chamorro, Cristina CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Álvarez, Rosa; Jimeno, M. Luisa CSIC ORCID; Martín Domenech, Angel; Pérez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Jan; San-Félix, Ana CSIC ORCID ; Camarasa Rius, María José CSIC ORCID | artículo |
| openAccess |  | 2015 | Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomers | Rivero-Buceta, Eva CSIC ORCID; Carrero, Paula CSIC; Casanova, Elena CSIC; Doyagüez, Elisa G. CSIC; Madrona, Andrés CSIC ORCID; Quesada, Ernesto CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Mateos, Raquel CSIC ORCID ; Bravo, Laura CSIC ORCID; Mathys, Leen; Noppen, Sam; Kiselev, Evgency; Marchand, Christophe; Pommier, Yves; Liekens, Sandra; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
| closedAccess |  | 2001 | Anti-HIV-1 activity of benzothiadiazine dioxide | Martínez Gil, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Castro, Ana CSIC ORCID; Pérez, Concepción CSIC ORCID; Witvrouw, M.; Pannecouque, C.; Balzarini, Jan; De Clercq, Erik | artículo |
| closedAccess |  | nov-2013 | Carbohydrate-binding agents act as potent trypanocidals that elicit modifications in VSG glycosylation and reduced virulence in Trypanosoma brucei | Castillo-Acosta, Victor M.; Vidal, Antonio E. CSIC ORCID ; Ruiz-Pérez, Luis Miguel; Van Damme, Els J. M.; Igarashi, Yasuhiro; Balzarini, Jan; González-Pacanowska, Dolores | artículo |
| openAccess |  | 23-sep-2016 | Carbohydrate-Binding Non-Peptidic Pradimicins for the Treatment of Acute Sleeping Sickness in Murine Models | Castillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Etxebarria, Juan; Reichardt, Niels Christian; Navarro, M.; Igarashi, Yasuhiro; Liekens, Sandra; Balzarini, Jan; González-Pacanowska, Dolores | artículo |
| openAccess |  | 2015 | Conservation of antiviral activity and improved selectivity in PMEO-DAPym upon pyrimidine to triazine scaffold hopping | Castro, Sonia de CSIC ORCID; Fernández-Cureses, Gloria CSIC; Andrei, G; Snoeck, R.; Sánchez-Murcia, Pedro A. CSIC ORCID; Korban, B.; Gago, Federico CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
| closedAccess | | 2011 | Crystal structure of tert -butyldimethylsilyl-spiroaminooxathioledioxide- thymine (TSAO-T) in complex with HIV-1 reverse transcriptase (RT) redefines the elastic limits of the non-nucleoside inhibitor-binding pocket | Das, Krishna; Bauman, J. D.; Rim, A. S.; Dharia, C.; Clark, A. D.; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Arnold, E. | artículo |
| openAccess |  | 2015 | Design, synthesis, and biological evaluation of unconventional aminopyrimidine, aminopurine, and amino-1,3,5-triazine methyloxynucleosides | Fernández-Cureses, Gloria CSIC; Castro, Sonia de CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
| closedAccess | | 2011 | Dipeptidyl peptidase IV dependent water-soluble prodrugs of highly lipophilic bicyclic nucleoside analogues | Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Andrei, G; Snoeck, R.; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess | | 2012 | Dipeptidyl Peptidase IV-Activated Prodrugs of Anti- Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer Systems | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 2015 | Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: A successful strategy for improving water solubility and oral bioavailability | Velázquez, Sonsoles CSIC ORCID CVN; Castro, Sonia de CSIC ORCID; Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
| closedAccess | | 3-feb-2012 | Dipeptidyl-peptidase IV (DPPIV/CD26)-based prodrugs of hydroxy-containing drugs | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; Lambeir, Anne-Marie; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess |  | 2014 | Discovery and SAR studies of a novel class of cytotoxic 1,4-disubstituted piperidines via Ugi reaction | Castro, Sonia de CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 6-mar-2015 | Exposure of Trypanosoma brucei to an N-acetylglucosamine-Binding Lectin Induces VSG Switching and Glycosylation Defects Resulting in Reduced Infectivity | Castillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Van Damme, Els J. M.; Balzarini, Jan; González-Pacanowska, Dolores | artículo |
| closedAccess |  | 2005 | From 1-acyl-β-lactam human cytomegalovirus protease inhibitors to 1-benzyloxycarbonylazetidines with improved antiviral activity. A straightforward approach to convert covalent to noncovalent inhibitors | Gerona-Navarro, Guillermo CSIC; Pérez de Vega, M. Jesús CSIC ORCID; García-López, M. Teresa CSIC ; Andrei, G; Snoeck, R.; Clercq, Erik De; Balzarini, Jan; González-Muñiz, Rosario CSIC ORCID | artículo |
| closedAccess | | 2011 | From β-Amino-γ-sultone to Unusual Bicyclic Pyridine and Pyrazine Heterocyclic Systems: Synthesis and Cytostatic and Antiviral Activities | Castro, Sonia de CSIC ORCID; Familiar, Olga CSIC; Andrei, G; Snoeck, R.; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 21-jul-2011 | gp120 -binding benzene compounds and saccharide compounds | Balzarini, Jan; Carrero, Paula CSIC; Casanova, Elena; Peréz-Pérez, María-Jesús CSIC ORCID ; San-Félix, Ana CSIC ORCID | solicitud de patente |
| closedAccess | | 2000 | HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique? | Camarasa Rius, María José CSIC ORCID; San-Felix, Alejandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; Chamorro, Cristina CSIC; Jimeno, M. Luisa CSIC ORCID; Perez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Jan | artículo |
| closedAccess |  | 2009 | Identification of aspartic acid-203 in human thymidine phosphorylase as an important residue for both catalysis and non-competitive inhibition by the small molecule >crystallization chaperone> 5′-O-tritylinosine (KIN59) | Bronckaers, A.; Aguado, Leire CSIC; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID ; Gago, Federico CSIC ORCID; Liekens, S. | artículo |
| openAccess |  | 12-mar-2009 | Improvements in or relating to compositions for the treatment or prophylaxis of viral infections | Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | patente |
