English   español  

Navegación por Autor rp00561

Ir a: 0-9 A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
O introducir las primeras letras:  
Mostrando resultados 27 a 46 de 70 < Anterior   Siguiente >
DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccessMascaraque Tet Lett2008_postprint.pdf.jpg2008Efficient one-pot synthesis of 1-alkoxy-2-arylaminoimidazolines from N-alkoxy-N-(2-aminoethyl)-2-nitrobenzenesulfonamides and arylisothiocyanatesMascaraque, Ainhoa CSIC; Nieto, Lidia CSIC; Dardonville, Christophe CSIC ORCID artículo
openAccess2004Fentanyl derivatives bearing aliphatic alkaneguanidinium moieties: A new series of hybrid molecules with significant binding affinity for μ-opioid receptors and I2-imidazoline binding sitesDardonville, Christophe CSIC ORCID ; Jagerovic, Nadine CSIC ORCID ; Callado, Luis F.; Meana, J. J.artículo
openAccessNucleic Acids Research, 2017,.pdf.jpg2017Functional and structural analysis of AT-specific minor groove binders that disrupt DNA-protein interactions and cause disintegration of the Trypanosoma brucei kinetoplastMillan, C. R.; Acosta-Reyes, F. J..; Lagartera, Laura CSIC ORCID; Ebiloma, Godwin U.; Lemgruber, L.; Nué Martínez, J. Jonathan CSIC ORCID; Saperas, Nuria CSIC ORCID; Dardonville, Christophe CSIC ORCID ; de Koning, Harry P.; Campos, J. Lourdesartículo
openAccess21-11489NP accepted mainmanuscript.pdf.jpg2021High yield synthesis of trans-Azoxybenzene versus 2-isopropoxy-4-nitrobenzoic acid: Influence of temperature and base concentrationNué Martínez, J. Jonathan CSIC ORCID; Alkorta, Ibon CSIC ORCID ; Dardonville, Christophe CSIC ORCID artículo
closedAccess2004Homoheteroaromaticity: the case study of azepine and dibenzazepineDardonville, Christophe CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; Alkorta, Ibon CSIC ORCID ; Elguero, José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2002I2-imidazoline binding site affinity of a structurally different type of ligandsDardonville, Christophe CSIC ORCID ; Rozas, Isabel; Callado, Luis F.; Meana, J. Javierartículo
closedAccessaccesoRestringido.pdf.jpg2004Imidazoline Binding Sites andTheir Ligands: An Overview of the Di¡erent Chemical StructuresDardonville, Christophe CSIC ORCID ; Rozas, Isabelartículo
openAccessacsmedchemlett.1c00717.pdf.jpg2022Imidazoline- and Benzamidine-Based Trypanosome Alternative Oxidase Inhibitors: Synthesis and Structure-Activity Relationship StudiesCisneros, David CSIC; Cueto-Díaz, Eduardo J. CSIC ORCID; Medina-Gil, T.; Chevillard, R.; Bernal-Fraile, T.; López-Sastre, R.; Aldfer, M. M.; Ungogo, M. A.; Elati, H. A. A.; Arai, N.; Otani, M.; Matsushiro, S.; Kojima, C.; Ebiloma, Godwin U.; Shiba, T.; De Koning, H. P.; Dardonville, Christophe CSIC ORCID artículo
openAccess2014In and out of the minor groove: Interaction of an AT-rich DNA with the drug CD27Acosta-Reyes, F. J..; Dardonville, Christophe CSIC ORCID ; de Koning, Harry P.; Natto, M.; Subirana, Juan A.; Campos, J. L.artículo
closedAccessaccesoRestringido.pdf.jpg2015Influence of ornithine decarboxylase antizymes and antizyme inhibitors on agmatine uptake by mammalian cellsRamos-Molina, Bruno; López-Contreras, Andrés J. CSIC ORCID; Lambertos, A.; Dardonville, Christophe CSIC ORCID ; Cremades, Asunción; Peñafiel, Rafaelartículo
openAccessES2668494A1.pdf.jpg18-may-2018Inhibidores alostéricos de TAO como agentes antiparasitarios y antifúngicosDardonville, Christophe CSIC ORCID ; Konning, Hendrik Pieter de; Ebiloma, Godwin U.solicitud de patente
openAccessES2668494B1.pdf.jpg16-may-2018Inhibidores alostéricos de TAO como agentes antiparasitarios y antifúngicosDardonville, Christophe CSIC ORCID ; Konning, Hendrik Pieter de; Ebiloma, Godwin U.patente
closedAccessaccesoRestringido.pdf.jpg2018Inhibition of trypanosome alternative oxidase without its N-terminal mitochondrial targeting signal (ΔMTS-TAO) by cationic and non-cationic 4-hydroxybenzoate and 4-alkoxybenzaldehyde derivatives active against T. brucei and T. congolenseEbiloma, Godwin U.; Díaz, Teresa; Balogun, Emmanuel O.; Abad, Lucía; Donachie, Anne; Kaiser, Marcel; Herraiz Tomico, Tomás CSIC ORCID ; Inaoka, Daniel K.; Shiba, Tomoo; Harada, Shigeharu; Kita, Kiyoshi; Koning, Harry P. de; Dardonville, Christophe CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2015Lowering the pK<inf>a</inf> of a bisimidazoline lead with halogen atoms results in improved activity and selectivity against Trypanosoma brucei in vitroRíos Martínez, Carlos H. CSIC; Nué Martínez, J. Jonathan CSIC ORCID; Ebiloma, Godwin U.; de Koning, Harry P.; Alkorta, Ibon CSIC ORCID ; Dardonville, Christophe CSIC ORCID artículo
openAccessBioorg. Med. Chem. Lett.pdf.jpg2022Methyl N-(tert-butoxycarbonyl)pyridine-2-carbimidothioate: A new reagent for the synthesis of N-phenylpyridinecarboxamidine (“arylimidamide”) DNA-minor groove binders from poorly nucleophilic aminesNué Martínez, J. Jonathan CSIC ORCID; Cisneros, David CSIC; Dardonville, Christophe CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg17-nov-2016Mitochondrion targeted trypanosome alternative oxidase inhibitors as chemotherapeutic agents against T. bruceiDardonville, Christophe CSIC ORCID ; Fueyo-González, Francisco CSIC ORCID; Díaz Ayuga, Teresa; Ebiloma, Godwin U.; Izquierdo García, C.; Bruggeman, V.; Sánchez Villamañán, J. M.; Donachie, Anne; Balogun, Emmanuel O.; Kita, Kiyoshi; Koning, Harry P. decomunicación de congreso
closedAccessjul-2000New aromatic iminoimidazolidine derivatives as alpha(1)-adrenoceptor antagonists: A novel synthetic approach and pharmacological activityDardonville, Christophe CSIC ORCID ; Goya, Pilar CSIC ORCID; Rozas, Isabel; Alsasua, Ángela; Martín, M. Isabel CSICartículo
closedAccessaccesoRestringido.pdf.jpg2000New aromatic iminoimidazolidine derivatives as α1-adrenoceptor antagonists: A novel synthetic approach and pharmacological activityDardonville, Christophe CSIC ORCID ; Goya, Pilar CSIC ORCID; Rozas, Isabel; Alsasua, Ángela; Martín, M. Isabel CSICartículo
Luque-Ortega JMC2010_postprint.pdf.jpg2010New Benzophenone-derived bisphosphonium salts as leishmanicidal leads targeting mitochondria through inhibition of respiratory complex IILuque-Ortega, Juan Román CSIC ORCID ; Reuther, Peter; Rivas, Luis CSIC ORCID ; Dardonville, Christophe CSIC ORCID artículo
Rodriguez et al JMC2008_postprint.pdf.jpg2008New bis(2-aminoimidazoline) and bisguanidine DNA minor groove binders with potent in vivo antitrypanosomal and antiplasmodial activityRodríguez, F. CSIC; Rozas, Isabel; Kaiser, M.; Brun, R.; Nguyen, Binh; Wilson, W. David; García, Rory Nelson; Dardonville, Christophe CSIC ORCID artículo