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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2008 | Efficient one-pot synthesis of 1-alkoxy-2-arylaminoimidazolines from N-alkoxy-N-(2-aminoethyl)-2-nitrobenzenesulfonamides and arylisothiocyanates | Mascaraque, Ainhoa CSIC; Nieto, Lidia CSIC; Dardonville, Christophe CSIC ORCID | artículo |
openAccess | | 2004 | Fentanyl derivatives bearing aliphatic alkaneguanidinium moieties: A new series of hybrid molecules with significant binding affinity for μ-opioid receptors and I2-imidazoline binding sites | Dardonville, Christophe CSIC ORCID ; Jagerovic, Nadine CSIC ORCID ; Callado, Luis F.; Meana, J. J. | artículo |
openAccess | | 2017 | Functional and structural analysis of AT-specific minor groove binders that disrupt DNA-protein interactions and cause disintegration of the Trypanosoma brucei kinetoplast | Millan, C. R.; Acosta-Reyes, F. J..; Lagartera, Laura CSIC ORCID; Ebiloma, Godwin U.; Lemgruber, L.; Nué Martínez, J. Jonathan CSIC ORCID; Saperas, Nuria CSIC ORCID; Dardonville, Christophe CSIC ORCID ; de Koning, Harry P.; Campos, J. Lourdes | artículo |
openAccess | | 2021 | High yield synthesis of trans-Azoxybenzene versus 2-isopropoxy-4-nitrobenzoic acid: Influence of temperature and base concentration | Nué Martínez, J. Jonathan CSIC ORCID; Alkorta, Ibon CSIC ORCID ; Dardonville, Christophe CSIC ORCID | artículo |
closedAccess | | 2004 | Homoheteroaromaticity: the case study of azepine and dibenzazepine | Dardonville, Christophe CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; Alkorta, Ibon CSIC ORCID ; Elguero, José CSIC ORCID | artículo |
closedAccess | | 2002 | I2-imidazoline binding site affinity of a structurally different type of ligands | Dardonville, Christophe CSIC ORCID ; Rozas, Isabel; Callado, Luis F.; Meana, J. Javier | artículo |
closedAccess | | 2004 | Imidazoline Binding Sites andTheir Ligands: An Overview of the Di¡erent Chemical Structures | Dardonville, Christophe CSIC ORCID ; Rozas, Isabel | artículo |
openAccess | | 2022 | Imidazoline- and Benzamidine-Based Trypanosome Alternative Oxidase Inhibitors: Synthesis and Structure-Activity Relationship Studies | Cisneros, David CSIC; Cueto-Díaz, Eduardo J. CSIC ORCID; Medina-Gil, T.; Chevillard, R.; Bernal-Fraile, T.; López-Sastre, R.; Aldfer, M. M.; Ungogo, M. A.; Elati, H. A. A.; Arai, N.; Otani, M.; Matsushiro, S.; Kojima, C.; Ebiloma, Godwin U.; Shiba, T.; De Koning, H. P.; Dardonville, Christophe CSIC ORCID | artículo |
openAccess | | 2014 | In and out of the minor groove: Interaction of an AT-rich DNA with the drug CD27 | Acosta-Reyes, F. J..; Dardonville, Christophe CSIC ORCID ; de Koning, Harry P.; Natto, M.; Subirana, Juan A.; Campos, J. L. | artículo |
closedAccess | | 2015 | Influence of ornithine decarboxylase antizymes and antizyme inhibitors on agmatine uptake by mammalian cells | Ramos-Molina, Bruno; López-Contreras, Andrés J. CSIC ORCID; Lambertos, A.; Dardonville, Christophe CSIC ORCID ; Cremades, Asunción; Peñafiel, Rafael | artículo |
openAccess | | 18-may-2018 | Inhibidores alostéricos de TAO como agentes antiparasitarios y antifúngicos | Dardonville, Christophe CSIC ORCID ; Konning, Hendrik Pieter de; Ebiloma, Godwin U. | solicitud de patente |
openAccess | | 16-may-2018 | Inhibidores alostéricos de TAO como agentes antiparasitarios y antifúngicos | Dardonville, Christophe CSIC ORCID ; Konning, Hendrik Pieter de; Ebiloma, Godwin U. | patente |
closedAccess | | 2018 | Inhibition of trypanosome alternative oxidase without its N-terminal mitochondrial targeting signal (ΔMTS-TAO) by cationic and non-cationic 4-hydroxybenzoate and 4-alkoxybenzaldehyde derivatives active against T. brucei and T. congolense | Ebiloma, Godwin U.; Díaz, Teresa; Balogun, Emmanuel O.; Abad, Lucía; Donachie, Anne; Kaiser, Marcel; Herraiz Tomico, Tomás CSIC ORCID ; Inaoka, Daniel K.; Shiba, Tomoo; Harada, Shigeharu; Kita, Kiyoshi; Koning, Harry P. de; Dardonville, Christophe CSIC ORCID | artículo |
closedAccess | | 2015 | Lowering the pK<inf>a</inf> of a bisimidazoline lead with halogen atoms results in improved activity and selectivity against Trypanosoma brucei in vitro | Ríos Martínez, Carlos H. CSIC; Nué Martínez, J. Jonathan CSIC ORCID; Ebiloma, Godwin U.; de Koning, Harry P.; Alkorta, Ibon CSIC ORCID ; Dardonville, Christophe CSIC ORCID | artículo |
openAccess | | 2022 | Methyl N-(tert-butoxycarbonyl)pyridine-2-carbimidothioate: A new reagent for the synthesis of N-phenylpyridinecarboxamidine (“arylimidamide”) DNA-minor groove binders from poorly nucleophilic amines | Nué Martínez, J. Jonathan CSIC ORCID; Cisneros, David CSIC; Dardonville, Christophe CSIC ORCID | artículo |
closedAccess | | 17-nov-2016 | Mitochondrion targeted trypanosome alternative oxidase inhibitors as chemotherapeutic agents against T. brucei | Dardonville, Christophe CSIC ORCID ; Fueyo-González, Francisco CSIC ORCID; Díaz Ayuga, Teresa; Ebiloma, Godwin U.; Izquierdo García, C.; Bruggeman, V.; Sánchez Villamañán, J. M.; Donachie, Anne; Balogun, Emmanuel O.; Kita, Kiyoshi; Koning, Harry P. de | comunicación de congreso |
closedAccess | | jul-2000 | New aromatic iminoimidazolidine derivatives as alpha(1)-adrenoceptor antagonists: A novel synthetic approach and pharmacological activity | Dardonville, Christophe CSIC ORCID ; Goya, Pilar CSIC ORCID; Rozas, Isabel; Alsasua, Ángela; Martín, M. Isabel CSIC | artículo |
closedAccess | | 2000 | New aromatic iminoimidazolidine derivatives as α1-adrenoceptor antagonists: A novel synthetic approach and pharmacological activity | Dardonville, Christophe CSIC ORCID ; Goya, Pilar CSIC ORCID; Rozas, Isabel; Alsasua, Ángela; Martín, M. Isabel CSIC | artículo |
| | 2010 | New Benzophenone-derived bisphosphonium salts as leishmanicidal leads targeting mitochondria through inhibition of respiratory complex II | Luque-Ortega, Juan Román CSIC ORCID ; Reuther, Peter; Rivas, Luis CSIC ORCID ; Dardonville, Christophe CSIC ORCID | artículo |
| | 2008 | New bis(2-aminoimidazoline) and bisguanidine DNA minor groove binders with potent in vivo antitrypanosomal and antiplasmodial activity | Rodríguez, F. CSIC; Rozas, Isabel; Kaiser, M.; Brun, R.; Nguyen, Binh; Wilson, W. David; García, Rory Nelson; Dardonville, Christophe CSIC ORCID | artículo |