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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccess2018Binding of eEF1A2 to the RNA-dependent protein kinase PKR modulates its activity and promotes tumour cell survivalLosada, Alejandro CSIC; Muñoz-Alonso, María J. CSIC; Martínez-Díez, Marta; Gago, Federico CSIC ORCID; Dominguez, Juan Manuel; Martínez-Leal, Juan Fernando; Galmarini, Carlos M.artículo
closedAccessaccesoRestringido.pdf.jpg2018Characterization of an atypical, thermostable, organic solvent- and acid-tolerant 2′-deoxyribosyltransferase from Chroococcidiopsis thermalisArco, J. del; Sánchez-Murcia, Pedro A. CSIC ORCID; Mancheño, Jose M. CSIC ORCID; Gago, Federico CSIC ORCID; Fernández-Lucas, J.artículo
openAccessene-2023Chemical modulation of microtubule structure as a tool to target different diseasesEstévez-Gallego, Juan CSIC ORCID ; Álvarez-Bernad, Beatriz CSIC; Lucena-Agell, Daniel CSIC ORCID ; Bonato, Francesca CSIC ORCID; Giménez-Abián, Juan F. CSIC ; Blanco, Óscar; París, Rebeca; Fuertes, L.; Martínez, J. C.; Kamimura, Shinji; Gago, Federico CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Oliva, María A. CSIC ORCID comunicación de congreso
openAccessStructure_Estévez-Gallego_2022.pdf.jpg5-ene-2023Chemical modulation of microtubule structure through the laulimalide/peloruside siteEstévez-Gallego, Juan CSIC ORCID ; Álvarez-Bernad, Beatriz CSIC; Benet, Pera; Wullschleger, Christoph; Raes, Olivier; Menche, Dirk; Martínez, Juan Carlos; Lucena-Agell, Daniel CSIC ORCID ; Prota, Andrea E.; Bonato, Francesca CSIC ORCID; Bargsten, Katja; Cornelus, Jelle; Giménez-Abián, Juan F. CSIC ; Northcote, Peter; Steinmetz, Michel O.; Kamimura, Shinji; Altmann, Karl-Heinz; Paterson, Ian; Gago, Federico CSIC ORCID; Van der Eycken, Johan; Díaz, José Fernando CSIC ORCID ; Oliva, María A. CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2019Cold-induced aldimine bond cleavage by Tris in: Bacillus subtilis alanine racemaseBernardo-García, Noelia CSIC; Sánchez-Murcia, Pedro A. CSIC ORCID; Espaillat, Akbar; Martínez-Caballero, Siseth ; Cava, Felipe CSIC ORCID; Hermoso, Juan A. CSIC ORCID; Gago, Federico CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2012Comparative Binding Energy (COMBINE) Analysis Supports a Proposal for the Binding Mode of Epothilones to β-TubulinCoderch, Claire; Klett, Javier CSIC ORCID; Morreale, Antonio; Díaz, José Fernando CSIC ORCID ; Gago, Federico CSIC ORCIDartículo
openAccessMJC-4.pdf.jpg2015Comparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductaseSánchez-Murcia, Pedro A. CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Toro, Miguel Ángel; Lucio, H. de; Jiménez, M. Angeles CSIC ORCID ; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccessaccesoRestringido.pdf.jpg2013Comparison of ultra-fast 2D and 3D ligand and target descriptors for side effect prediction and network analysis in polypharmacologyCortés Cabrera, Álvaro CSIC ORCID; Morris, Garret M.; Finn, Paul W.; Morreale, Antonio; Gago, Federico CSIC ORCIDartículo
openAccessmarinedrugs-21-00100-v2.pdf.jpg2023Computational Approaches to Enzyme Inhibition by Marine Natural Products in the Search for New DrugsGago, Federico CSIC ORCIDartículo de revisión
openAccessMJC-1.pdf.jpg2015Conservation of antiviral activity and improved selectivity in PMEO-DAPym upon pyrimidine to triazine scaffold hoppingCastro, Sonia de CSIC ORCID; Fernández-Cureses, Gloria CSIC; Andrei, G; Snoeck, R.; Sánchez-Murcia, Pedro A. CSIC ORCID; Korban, B.; Gago, Federico CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2012CRDOCK: An ultrafast multipurpose protein-ligand docking toolCortés Cabrera, Álvaro CSIC ORCID; Klett, Javier CSIC ORCID; Dos Santos, Helena G.; Perona, Almudena CSIC ORCID CVN; Gil Redondo, Rubén; Francis, Sandrea M. CSIC; Priego, Eva María CSIC ORCID; Gago, Federico CSIC ORCID; Morreale, Antonioartículo
openAccess2341603_B1.pdf.jpg28-abr-2011Derivados de nucleósidos para el tratamiento de infecciones por LeishmaniaGago, Federico CSIC ORCID; Rico Galán, Eva; Camarasa Rius, María José CSIC ORCID; Jiménez, A. R.; Casanova Malpica, Elena; Moreno Mateos, David; Peréz-Pérez, María-Jesús CSIC ORCID patente
openAccessJ. AM. CHEM. SOC. 2003, 125, 16243-16260.pdf.jpg2003Development of a new family of conformationally restricted peptides as potent nucleators of β-turns. Design, synthesis, structure, and biological evaluation of a β-lactam peptide analogue of melanostatinPalomo, Claudio; Aizpurua, Jesús M.; Benito, Ana M. ; Miranda, José Ignacio; Fratila, Raluca M. CSIC ORCID; Matute, Carlos; Domercq, Maria; Gago, Federico CSIC ORCID; Martin-Santamaria, Sonsoles; Linden, Anthonyartículo
openAccessja038180asi20031002_103725.pdf.jpg2003Development of a new family of conformationally restricted peptides as potent nucleators of β-turns. Design, synthesis, structure, and biological evaluation of a β-lactam peptide analogue of melanostatin. Supporting InformationPalomo, Claudio; Aizpurua, Jesús M.; Benito, Ana M. ; Miranda, José Ignacio; Fratila, Raluca M. CSIC ORCID; Matute, Carlos; Domercq, Maria; Gago, Federico CSIC ORCID; Martin-Santamaria, Sonsoles; Linden, Anthonydataset
openAccess2006Discovery of TSAO derivatives with an unusual HIV-1 activity/resistance profileCastro, Sonia de CSIC ORCID ; García-Aparicio, Carlos CSIC; Van Laethem, K.; Gago, Federico CSIC ORCID; Lobatón, E.; De Clercq, E.; Balzarini, J.; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccessaccesoRestringido.pdf.jpg2020Distinct binding of cetirizine enantiomers to human serum albumin and the human histamine receptor H1Perona, Almudena CSIC ORCID CVN; Ros, M. Piedad; Mills, Alberto; Morreale, Antonio; Gago, Federico CSIC ORCIDartículo
openAccessacs.jmedchem.1c00315-1.pdf.jpg7-jul-2021Double Arylation of the Indole Side Chain of Tri- and Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV‑1 and EV-A71 Entry InhibitorsMartí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Puente-Secades, Sofía de la CSIC; Mills, Alberto; Quesada, Ernesto CSIC ORCID ; Abdelnabi, Rana; Sun, Liang; Boonen, Arnaud; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
openAccessacs.jmedchem.1c00206.pdf.jpg2021Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazolesRevuelto, Alejandro CSIC ORCID; Lucio, Héctor de; García-Soriano, Juan Carlos; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessenantioselective_oxidation_benavente.pdf.jpg2015Enantioselective oxidation of galactitol 1-phosphate by galactitol-1-phosphate 5-dehydrogenase from Escherichia coliBenavente, Rocio CSIC; Esteban-Torres, María CSIC ORCID; Kohring, G. W.; Cortés Cabrera, Álvaro CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Acebrón, Iván CSIC ORCID; Rivas, Blanca de las CSIC ORCID; Muñoz, Rosario CSIC ORCID ; Mancheño, Jose M. CSIC ORCIDartículo
openAccess734083.pdf.jpg18-jul-2018Enzymatic synthesis of therapeutic nucleosides using a highly versatile purine nucleoside 2’-Deoxyribosyl transferase from Trypanosoma bruceiPérez, Elena; Sánchez-Murcia, Pedro A. CSIC ORCID; Jordaan, Justin; Blanco, María Dolores; Mancheño, Jose M. CSIC ORCID; Gago, Federico CSIC ORCID; Fernández-Lucas, J.artículo