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Browsing by Author De Clercq, Erik

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Showing results 1 to 19 of 19
RightsPreviewIssue DateTitleAuthor(s)Type
closedAccessaccesoRestringido.pdf.jpg18-Jun-20185-Hydroxypyrido[2,3-b]pyrazin-6(5H)-one derivatives as novel dual inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H and integraseSun, Lin; Gao, Ping; Dong, Guanyu; Zhang, Xujie; Ding, Xiao; Wang, Xueshun; Daelemans, Dirk; De Clercq, Erik; Pannecouque, Christophe; Menéndez-Arias, Luis CSIC ORCID ; Zhang, Peng; Liu, Xinyongartículo
closedAccess1998Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptaseVelázquez, Sonsoles CSIC ORCID CVN; Chamorro, Cristina CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Álvarez, Rosa; Jimeno, M. Luisa CSIC ORCID; Martín Domenech, Angel; Pérez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Jan; San-Félix, Ana CSIC ORCID ; Camarasa Rius, María José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpgFeb-1993Activity of several S-adenosylhomocysteine hydrolase inhibitors against African swine fever virus replication in Vero cellsVillalón, M.; Gil-Fernández, Carmen ; De Clercq, Erikartículo
closedAccessArtículo.pdf.jpg2001Anti-HIV-1 activity of benzothiadiazine dioxideMartínez Gil, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Castro, Ana CSIC ORCID; Pérez, Concepción CSIC ORCID; Witvrouw, M.; Pannecouque, C.; Balzarini, Jan; De Clercq, Erikartículo
openAccess340989_Manuscript-revised_LMA_Gao0702_LMA.pdf.jpg1-Sep-2019Design, synthesis and biological evaluation of 3-hydroxyquinazoline-2,4(1H,3H)-diones as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and integraseGao, Ping; Cheng, Xiqiang; Sun, Lin; Song, Shu; Álvarez, Mar CSIC ORCID; Luczkowiak, Joanna; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Peng; Liu, Xinyongartículo
openAccessMenéndez-AriasL_DesignSynthesisandBiologic.pdf.jpg24-Nov-2018Design, synthesis, and biologic evaluation of novel galloyl derivatives as HIV-1 RNase H inhibitorsGao, Ping; Sun, Lin; Cheng, Xiqiang; Poongavanam, Vasanthanathan; Kongsted, Jacob; Álvarez, Mar CSIC ORCID; Luczkowiak, Joanna; Pannecouque, Christophe; De Clercq, Erik; Lee, Kuo-Hsiung; Chen, Chin-Ho; Liu, Huiqing; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhang, Pengartículo
openAccessMenéndez-AriasL_DiscoveryOptimizationAndTarget.pdf.jpg2021Discovery, optimization, and target identification of novel coumarin derivatives as HIV-1 reverse transcriptase-associated ribonuclease H inhibitorsKang, Dongwei; Urhan, Çagil; Wei, Fenju; Frutos-Beltrán, Estrella CSIC ORCID; Sun, Lin; Álvarez, Mar CSIC ORCID; Feng, Da; Tao, Yucen; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo
closedAccess2000HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique?Camarasa Rius, María José CSIC ORCID; San-Felix, Alejandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; Chamorro, Cristina CSIC; Jimeno, M. Luisa CSIC ORCID; Perez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Janartículo
openAccessMenéndez-AriasL_MedicinalChemistryStrategies.pdf.jpg17-Feb-2021Medicinal chemistry strategies for discovering antivirals effective against drug-resistant virusesMa, Yue; Frutos-Beltrán, Estrella CSIC ORCID; Kang, Dongwei; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo de revisión
openAccessMenéndez-AriasL_MedicinalChemistryStrategies.pdf.jpg17-Feb-2021Medicinal chemistry strategies for discovering antivirals effective against drug-resistant virusesMa, Yue; Frutos-Beltrán, Estrella CSIC ORCID; Kang, Dongwei; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo de revisión
openAccessMenéndez-AriasL_MedicinalChemistryStrategies.pdf.jpg17-Feb-2021Medicinal chemistry strategies for discovering antivirals effective against drug-resistant virusesMa, Yue; Frutos-Beltrán, Estrella CSIC ORCID; Kang, Dongwei; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo de revisión
closedAccessaccesoRestringido.pdf.jpg2000Nonnucleoside human cytomegalovirus inhibitors: Synthesis and antiviral evaluation of (chlorophenylmethyl)benzothiadiazine dioxide derivativesMartínez Gil, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Pérez, Concepción CSIC ORCID; Castro, Ana CSIC ORCID; Prieto, Columbiana; Otero, Joaquín; Andrei, G; Snoeck, R.; Balzarini, Jan; De Clercq, Erikartículo
closedAccess1997Novel analogues of the anti HIV-1 agent TSAO-T modified at the 3'-spiro moietyÁlvarez, Rosa; Jimeno, M. Luisa CSIC ORCID; De Clercq, Erik; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
openAccessMenéndezAriasL_NovelIndolylarylsulfonederivatives.pdf.jpg12-Oct-2020Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181CGao, Ping; Song, Shu; Frutos-Beltrán, Estrella CSIC ORCID; Li, Wenxin; Sun, Bin; Kang, Dongwei; Zou, Jinmi; Zhang, Jian; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Peng; Liu, Xinyongartículo
closedAccess1999Potential multifunctional inhibitors of HIV-1 reverse transcriptase. Novel [AZT]-[TSAO-T] and [d4T]-[TSAO-T] heterodimers modified in the linker and in the dideoxynucleoside regionVelázquez, Sonsoles CSIC ORCID CVN; Tuñón, Victoria; Jimeno, M. Luisa CSIC ORCID; Chamorro, Cristina CSIC; De Clercq, Erik; Balzarini, Jan; Camarasa, María Joséartículo
closedAccessaccesoRestringido.pdf.jpg2001Second generation of TSAO compounds directed against HIV-1 TSAO-resistant strainsLobaton, E.; Velázquez, Sonsoles CSIC ORCID CVN; Peréz-Pérez, María-Jesús CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; San-Felix, S.; De Clercq, Erik; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess1995Synthesis and Anti-HIV Activity of [UT]-[TSAO-TI and [UT]-[HEPT] Dimers as Potential Multifunctional Inhibitors of HIV-1 Reverse TranscriptaseVelázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; San-Félix, Ana CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; De Clercq, Erik; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess1998Synthesis and anti-HIV properties of 1,2,4,6-thiatriazin-3-one 1,1-dioxide nucleosidesOchoa, Carmen; Provencio, Rafael; Jimeno, M. Luisa CSIC ORCID; Balzarini, Jan; De Clercq, Erikartículo
closedAccess1997Synthesis and anti-human immunodeficiency virus type 1 activity of novel 3'-spiro nucleoside analogues of TSAO-TÁlvarez, Rosa; Jimeno, M. Luisa CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; De Clercq, Erik; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo